Evidence map›Paper›PMID 40665896›Full record

ArticleCPT: pharmacometrics & systems pharmacology2025

From In Vitro Efficacy to Long-Term HbA1c Response for GLP-1R/GlucagonR Agonism Using the 4GI-HbA1c Systems Model.

Rolien Bosch, Marcella Petrone, Rosalin Arends, Eric J G Sijbrands, Sven Hoefman, Nelleke Snelder

Abstract read
In one paragraph

Article in CPT: pharmacometrics & systems pharmacology, 2025. The graph could read no effect estimate from its abstract, so it casts no vote on the map. Cited by 1 paper.

0numbers the graph read from it
0cells of the map it votes in
1citing papers in PubMed
–field-weighted citation impact
1 · What the graph read from it

What it found

Each row is one number read from the abstract, on the scale the paper reported it, with its interval. Left of the dashed line favours the treatment, right favours the comparator. Under each row is the sentence it came from. New to these charts? A ten-minute tutorial.

The abstract states no effect estimate the extractor could read, or names no intervention and outcome on the map, so this paper lights no cell and moves no belief. It is still indexed, cited and linked below.

2 · The registry

The trial behind it

Trials whose registry record cites this paper, or whose number appears in the abstract. A trial that started after this paper was published is citing it as background, not reporting it.

Neither the registry nor the abstract names a trial number. If this is a trial report, that itself is worth knowing.

3 · Its place in the literature

Who cites it

1 citing paper in PubMed.

  1. Article
4 · The record

Corrections and comments

PubMed lists nothing against this paper. Absence here is not a guarantee, only a check that was made.

5 · Who and what money

Authors and funding

6 authors.

Rolien BoschLAP&P Consultants, Leiden, the Netherlands.ORCID 0000-0002-6675-8303
Marcella PetroneClinical Pharmacology and Safety Sciences, AstraZeneca, Cambridge, UK.
Rosalin ArendsAstraZeneca, Gaithersburg, Maryland, USA.
Eric J G SijbrandsDepartment of Internal Medicine, Erasmus MC, University Medical Centre, Rotterdam, the Netherlands.ORCID 0000-0001-8857-7389
Sven HoefmanLAP&P Consultants, Leiden, the Netherlands.
Nelleke SnelderLAP&P Consultants, Leiden, the Netherlands.ORCID 0000-0003-1302-678X

Funding

No grant is acknowledged in the PubMed record.

6 · The paper itself

Abstract

For the treatment of Type 2 Diabetes, high efficacy approaches such as Glucagon-like peptide 1 (GLP-1)-based therapies are recommended for glucose control. Prediction of the clinical outcome of these therapies on glucose and hemoglobin A1c (HbA1c), using early available pharmacokinetic and in vitro efficacy information, can be a valuable tool for compound selection and supporting drug development. Our previously developed glucose homeostasis model (the 4GI model) is a systems model that is able to quantify drug effects on glucose based on in vitro potency and PK information. In this research, the model was coupled to an existing integrated glucose-red blood cell-HbA1c (IGRH) model for predicting the effects of GLP-1 and GLP-1/glucagon (dual) receptor agonists, liraglutide and cotadutide, on glucose and HbA1c. The 4GI model was validated for predicting 24-h glucose (C

Indexed as

Diabetes Mellitus, Type 2Glucagon-Like Peptide-1 Receptor AgonistsGlycated HemoglobinHypoglycemic AgentsModels, BiologicalReceptors, GlucagonBlood GlucoseGlucagon-Like Peptide-1 ReceptorHumansLiraglutideBlood GlucoseGLP1R protein, humanGlucagon-Like Peptide-1 ReceptorGlucagon-Like Peptide-1 Receptor AgonistsGlycated Hemoglobinhemoglobin A1c protein, humanHypoglycemic AgentsLiraglutideReceptors, Glucagon4GIcotadutidediabetesGLP‐1R agonistsQSPsystems pharmacology

Identifiers

PMID40665896
PMCPMC12439278

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Registered trials

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Read under generation 80e0d062 · epoch 390. Bibliography from PubMed, PubMed Central and OpenAlex; grants from NIH RePORTER; trial links from ClinicalTrials.gov; estimates, votes and beliefs from the OpenQuestion graph.