Evidence map›Paper›PMID 36548658›Full record

ArticleTropical medicine and infectious disease2022

A Novel Protocol for the Synthesis of 1,2,4-Oxadiazoles Active against Trypanosomatids and Drug-Resistant Leukemia Cell Lines.

Paulo Pitasse-Santos, Eduardo Salustiano, Raynná Bittencourt Pena, Otávio Augusto Chaves, Leonardo Marques da Fonseca, Kelli Monteiro da Costa, Carlos Antônio do Nascimento Santos, Jhenifer Santos Dos Reis, Marcos André Rodrigues da Costa Santos, Jose Osvaldo Previato and 7 more

Open access · goldAbstract read
In one paragraph

Article in Tropical medicine and infectious disease, 2022. The graph could read no effect estimate from its abstract, so it casts no vote on the map. Cited by 2 papers.

0numbers the graph read from it
0cells of the map it votes in
2citing papers in PubMed
0.4field-weighted citation impact, top 43% of its field
1 · What the graph read from it

What it found

Each row is one number read from the abstract, on the scale the paper reported it, with its interval. Left of the dashed line favours the treatment, right favours the comparator. Under each row is the sentence it came from. New to these charts? A ten-minute tutorial.

The abstract states no effect estimate the extractor could read, or names no intervention and outcome on the map, so this paper lights no cell and moves no belief. It is still indexed, cited and linked below.

2 · The registry

The trial behind it

Trials whose registry record cites this paper, or whose number appears in the abstract. A trial that started after this paper was published is citing it as background, not reporting it.

Neither the registry nor the abstract names a trial number. If this is a trial report, that itself is worth knowing.

3 · Its place in the literature

Who cites it

2 citing papers in PubMed, 4 citations in OpenAlex.

  1. Article
  2. Advancement in Leishmaniasis Diagnosis and Therapeutics.Tropical medicine and infectious disease · 2023
    Article
4 · The record

Corrections and comments

PubMed lists nothing against this paper. Absence here is not a guarantee, only a check that was made.

5 · Who and what money

Authors and funding

17 authors at 3 institutions in 2 countries.

Paulo Pitasse-SantosInstituto de Química, Universidade Federal Rural do Rio de Janeiro, Seropédica 23890-000, Rio de Janeiro, Brazil.
Eduardo SalustianoInstituto de Biofísica Carlos Chagas Filho, Universidade Federal do Rio de Janeiro, Rio de Janeiro 21491-170, Rio de Janeiro, Brazil.ORCID 0000-0001-5572-6130
Raynná Bittencourt PenaLaboratório Integrado de Computação Científica (LICC), Universidade Federal do Rio de Janeiro-Centro Multidisciplinar UFRJ Macaé, Macaé 27930-560, Rio de Janeiro, Brazil.
Otávio Augusto ChavesLaboratório de Imunofarmacologia, Instituto Oswaldo Cruz (IOC), Fundação Oswaldo Cruz (Fiocruz), Rio de Janeiro 21040-900, Rio de Janeiro, Brazil.ORCID 0000-0001-6211-7659
Leonardo Marques da FonsecaInstituto de Biofísica Carlos Chagas Filho, Universidade Federal do Rio de Janeiro, Rio de Janeiro 21491-170, Rio de Janeiro, Brazil.ORCID 0000-0001-8239-6843
Kelli Monteiro da CostaInstituto de Biofísica Carlos Chagas Filho, Universidade Federal do Rio de Janeiro, Rio de Janeiro 21491-170, Rio de Janeiro, Brazil.ORCID 0000-0001-6178-0942
Carlos Antônio do Nascimento SantosInstituto de Biofísica Carlos Chagas Filho, Universidade Federal do Rio de Janeiro, Rio de Janeiro 21491-170, Rio de Janeiro, Brazil.
Jhenifer Santos Dos ReisInstituto de Biofísica Carlos Chagas Filho, Universidade Federal do Rio de Janeiro, Rio de Janeiro 21491-170, Rio de Janeiro, Brazil.
Marcos André Rodrigues da Costa SantosInstituto de Biofísica Carlos Chagas Filho, Universidade Federal do Rio de Janeiro, Rio de Janeiro 21491-170, Rio de Janeiro, Brazil.
Jose Osvaldo PreviatoInstituto de Biofísica Carlos Chagas Filho, Universidade Federal do Rio de Janeiro, Rio de Janeiro 21491-170, Rio de Janeiro, Brazil.
Lucia Mendonça PreviatoInstituto de Biofísica Carlos Chagas Filho, Universidade Federal do Rio de Janeiro, Rio de Janeiro 21491-170, Rio de Janeiro, Brazil.ORCID 0000-0003-3927-3244
Leonardo Freire-de-LimaInstituto de Biofísica Carlos Chagas Filho, Universidade Federal do Rio de Janeiro, Rio de Janeiro 21491-170, Rio de Janeiro, Brazil.ORCID 0000-0003-3013-3173
Nelilma Correia RomeiroLaboratório Integrado de Computação Científica (LICC), Universidade Federal do Rio de Janeiro-Centro Multidisciplinar UFRJ Macaé, Macaé 27930-560, Rio de Janeiro, Brazil.
Lúcia Helena Pinto-da-SilvaInstituto de Veterinária, Universidade Federal Rural do Rio de Janeiro, Seropédica 23890-000, Rio de Janeiro, Brazil.
Célio G Freire-de-LimaInstituto de Biofísica Carlos Chagas Filho, Universidade Federal do Rio de Janeiro, Rio de Janeiro 21491-170, Rio de Janeiro, Brazil.ORCID 0000-0002-4148-3657
Débora Decotè-RicardoInstituto de Veterinária, Universidade Federal Rural do Rio de Janeiro, Seropédica 23890-000, Rio de Janeiro, Brazil.
Marco Edilson Freire-de-LimaInstituto de Química, Universidade Federal Rural do Rio de Janeiro, Seropédica 23890-000, Rio de Janeiro, Brazil.ORCID 0000-0003-0563-3483
Universidade Federal do Rio de Janeiro · BRUniversidade Federal Rural do Rio de Janeiro · BRFundação Oswaldo Cruz · BR

Funding

Conselho Nacional de Desenvolvimento e Pesquisa (CNPq)Fundação Carlos Chagas Filho de Amparo à Pesquisa do Estado do Rio de Janeiro (FAPERJ).the Brazilian agencies: Coordenação de Aperfeiçoamento de Pessoal de Nível Superior (CAPES) 001
6 · The paper itself

Abstract

Cancer and parasitic diseases, such as leishmaniasis and Chagas disease, share similarities that allow the co-development of new antiproliferative agents as a strategy to quickly track the discovery of new drugs. This strategy is especially interesting regarding tropical neglected diseases, for which chemotherapeutic alternatives are extremely outdated. We designed a series of (

Indexed as

anticancerchagas diseasechronic myeloid leukemiaLeishmania amazonensismolecular dockingTrypanosoma cruzi

Identifiers

PMID36548658
PMCPMC9787607
OpenAlexW4310143453

What OpenQuestion holds

Textmetadata
LicenceCC BY
Read underepoch 390

Registered trials

None linked

Read under generation 80e0d062 · epoch 390. Bibliography from PubMed, PubMed Central and OpenAlex; grants from NIH RePORTER; trial links from ClinicalTrials.gov; estimates, votes and beliefs from the OpenQuestion graph.