ArticleAngewandte Chemie (International ed. in English)2022
Borylation Directed Borylation of Indoles Using Pyrazabole Electrophiles: A One-Pot Route to C7-Borylated-Indolines.
Article in Angewandte Chemie (International ed. in English), 2022. The graph could read no effect estimate from its abstract, so it casts no vote on the map. Cited by 9 papers.
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Who cites it
9 citing papers in PubMed.
- Design, Synthesis, and Applications of Pyrazabole Functionalized Derivatives.Chemistry, an Asian journal · 2026Review
- Palladium-Catalyzed Heteroannulation of Bdan-Capped Alkynes: Rapid Access to Complex Indole Scaffolds.The Journal of organic chemistry · 2025Article
- Intermolecular SpAngewandte Chemie (International ed. in English) · 2025Article
- Borylation-Reduction-Borylation for the Formation of 1,4-Azaborines.Organic letters · 2023Article
- Borylation directed borylation ofChemical science · 2023Article
- Metal-free C-H Borylation and Hydroboration of Indoles.ACS omega · 2023Review
- Amides as modifiable directing groups in electrophilic borylation.Chemical science · 2023Article
- Synthesis of Electrophiles Derived from Dimeric Aminoboranes and Assessing Their Utility in the Borylation of π Nucleophiles.Organometallics · 2022Article
- Borylation Directed Borylation of Indoles Using Pyrazabole Electrophiles: A One-Pot Route to C7-Borylated-Indolines.Angewandte Chemie (International ed. in English) · 2022Article
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Authors and funding
5 authors.
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Abstract
Pyrazabole (1) is a readily accessible diboron compound that can be transformed into ditopic electrophiles. In 1 (and derivatives), the B⋅⋅⋅B separation is ca. 3 Å, appropriate for one boron centre bonding to N and one to the C7 of indoles and indolines. This suitable B⋅⋅⋅B separation enables double E-H (E=N/C) functionalisation of indoles and indolines. Specifically, the activation of 1 with HNTf
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