Evidence map›Paper›PMID 34948408›Full record

ArticleInternational journal of molecular sciences2021

Benzimidazole Derivatives as New and Selective Inhibitors of Arginase from

Irene Betancourt-Conde, Claudia Avitia-Domínguez, Alicia Hernández-Campos, Rafael Castillo, Lilián Yépez-Mulia, Jesús Oria-Hernández, Sara T Méndez, Erick Sierra-Campos, Mónica Valdez-Solana, Siseth Martínez-Caballero and 3 more

Open access · goldAbstract read
In one paragraph

Article in International journal of molecular sciences, 2021. The graph could read no effect estimate from its abstract, so it casts no vote on the map. Cited by 7 papers.

0numbers the graph read from it
0cells of the map it votes in
7citing papers in PubMed
1.2field-weighted citation impact, top 20% of its field
1 · What the graph read from it

What it found

Each row is one number read from the abstract, on the scale the paper reported it, with its interval. Left of the dashed line favours the treatment, right favours the comparator. Under each row is the sentence it came from. New to these charts? A ten-minute tutorial.

The abstract states no effect estimate the extractor could read, or names no intervention and outcome on the map, so this paper lights no cell and moves no belief. It is still indexed, cited and linked below.

2 · The registry

The trial behind it

Trials whose registry record cites this paper, or whose number appears in the abstract. A trial that started after this paper was published is citing it as background, not reporting it.

Neither the registry nor the abstract names a trial number. If this is a trial report, that itself is worth knowing.

3 · Its place in the literature

Who cites it

7 citing papers in PubMed, 11 citations in OpenAlex.

  1. Review
  2. Article
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  6. Recent Advances: Heterocycles in Drugs and Drug Discovery.International journal of molecular sciences · 2024
    Article
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4 · The record

Corrections and comments

PubMed lists nothing against this paper. Absence here is not a guarantee, only a check that was made.

5 · Who and what money

Authors and funding

13 authors at 6 institutions in 2 countries.

Irene Betancourt-CondeFacultad de Medicina y Nutrición, Universidad Juárez del Estado de Durango, Av. Universidad y Fanny Anitúa S/N, Durango 34000, Mexico.
Claudia Avitia-DomínguezFacultad de Medicina y Nutrición, Universidad Juárez del Estado de Durango, Av. Universidad y Fanny Anitúa S/N, Durango 34000, Mexico.
Alicia Hernández-CamposDepartamento de Farmacia, Facultad de Química, Universidad Nacional Autónoma de México, Mexico City 04510, Mexico.
Rafael CastilloDepartamento de Farmacia, Facultad de Química, Universidad Nacional Autónoma de México, Mexico City 04510, Mexico.
Lilián Yépez-MuliaUnidad de Investigación Médica en Enfermedades Infecciosas y Parasitarias, Unidad Médica de Alta Especialidad-Hospital de Pediatría, Centro Médico Nacional Siglo XXI, Instituto Mexicano del Seguro Social, Mexico City 06720, Mexico.ORCID 0000-0001-8675-5671
Jesús Oria-HernándezLaboratorio de Bioquímica-Genética, Instituto Nacional de Pediatría, Secretaría de Salud, Mexico City 04530, Mexico.ORCID 0000-0001-7147-1879
Sara T MéndezLaboratorio de Bioquímica-Genética, Instituto Nacional de Pediatría, Secretaría de Salud, Mexico City 04530, Mexico.ORCID 0000-0001-8619-1220
Erick Sierra-CamposFacultad de Ciencias Químicas, Universidad Juárez del Estado de Durango, Av. Artículo 123 S/N Fracc. Filadelfia, Gómez Palacio 35010, Mexico.ORCID 0000-0001-8622-4045
Mónica Valdez-SolanaFacultad de Ciencias Químicas, Universidad Juárez del Estado de Durango, Av. Artículo 123 S/N Fracc. Filadelfia, Gómez Palacio 35010, Mexico.
Siseth Martínez-CaballeroDepartamento de Cristalografía y Biología Estructural, Instituto Química-Física Rocasolano, Consejo Superior de Investigaciones Científicas, 28006 Madrid, Spain.
Juan A HermosoDepartamento de Cristalografía y Biología Estructural, Instituto Química-Física Rocasolano, Consejo Superior de Investigaciones Científicas, 28006 Madrid, Spain.
Antonio Romo-MancillasLaboratorio de Diseño Asistido por Computadora y Síntesis de Fármacos, Facultad de Química, Universidad Autónoma de Querétaro, Querétaro 76010, Mexico.ORCID 0000-0003-2869-588X
Alfredo Téllez-ValenciaFacultad de Medicina y Nutrición, Universidad Juárez del Estado de Durango, Av. Universidad y Fanny Anitúa S/N, Durango 34000, Mexico.ORCID 0000-0001-7629-4111
Universidad Juárez del Estado de Durango · MXConsejo Superior de Investigaciones Científicas · ESSecretaria de Salud · MXUniversidad Nacional Autónoma de México · MXAutonomous University of Queretaro · MXMexican Social Security Institute · MX

Funding

Consejo Nacional de Ciencia y Tecnología 257848, 258694Spanish Ministry of Science, Innovation and Competitiveness PID2020-115331GB-100
6 · The paper itself

Abstract

Leishmaniasis is a disease caused by parasites of the

Indexed as

AnimalsAntiprotozoal AgentsArginaseBenzimidazolesCell LineDrug DiscoveryHumansLeishmania mexicanaLeishmaniasis, CutaneousMiceModels, MolecularProtozoan ProteinsAntiprotozoal AgentsArginaseBenzimidazolesProtozoan Proteinsarginasebenzimidazole derivativesenzyme inhibitionleishmaniasismolecular dynamicsvirtual screening

Identifiers

PMID34948408
PMCPMC8705706
OpenAlexW4200469571

What OpenQuestion holds

Textmetadata
LicenceCC BY
Read underepoch 390

Registered trials

None linked

Read under generation 80e0d062 · epoch 390. Bibliography from PubMed, PubMed Central and OpenAlex; grants from NIH RePORTER; trial links from ClinicalTrials.gov; estimates, votes and beliefs from the OpenQuestion graph.