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ArticleBioorganic & medicinal chemistry2018

Synthesis and profiling of a 3-aminopyridin-2-one-based kinase targeted fragment library: Identification of 3-amino-5-(pyridin-4-yl)pyridin-2(1H)-one scaffold for monopolar spindle 1 (MPS1) and Aurora kinases inhibition.

Daren Fearon et al.PubMed ↗Full text ↗Publisher ↗

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