ArticleOrganic letters2012
Intramolecular Pd(II)-catalyzed aerobic oxidative amination of alkenes: synthesis of six-membered N-heterocycles.
Article in Organic letters, 2012. The graph could read no effect estimate from its abstract, so it casts no vote on the map. Cited by 18 papers.
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Who cites it
18 citing papers in PubMed.
- Rational drug design and synthesis of novel bioactive molecules with oxygen heterocycles, including AChE and BChE inhibitory properties and SAR studies.Molecular diversity · 2026Review
- Access to Fused Indolines with a QuaternaryOrganic letters · 2026Article
- Advances in Piperazine-based Compounds for Antimicrobial Drug Development: Design, SAR, and Therapeutic Potential.Current drug research reviews · 2026Review
- Competing Mechanisms in Palladium-Catalyzed Alkoxycarbonylation of Styrene.ACS catalysis · 2024Article
- Syntheses of 2- and 3-Substituted Morpholine Congeners via Ring Opening of 2-Tosyl-1,2-Oxazetidine.The Journal of organic chemistry · 2023Article
- Lewis Acid-Catalyzed Halonium Generation for Morpholine Synthesis and Claisen Rearrangement.The Journal of organic chemistry · 2022Article
- Oxidative Cyclization of Sulfamates onto Pendant Alkenes.Organic letters · 2020Article
- Synthesis of Indolines and Derivatives by Aza-Heck Cyclization.Angewandte Chemie (International ed. in English) · 2019Article
- A 5 + 1 Protic Acid Assisted Aza-Pummerer Approach for Synthesis of 4-Chloropiperidines from Homoallylic Amines.The Journal of organic chemistry · 2019Article
- Expedient syntheses of N-heterocycles via intermolecular amphoteric diamination of allenes.Nature communications · 2018Article
- Molecular ligand modulation of palladium nanocatalysts for highly efficient and robust heterogeneous oxidation of cyclohexenone to phenol.Science advances · 2017Article
- Diazafluorenone-Promoted Oxidation Catalysis: Insights into the Role of Bidentate Ligands in Pd-Catalyzed Aerobic Aza-Wacker Reactions.ACS catalysis · 2016Article
- Palladium-Catalyzed Modular Synthesis of Substituted Piperazines and Related Nitrogen Heterocycles.Organic letters · 2016Article
- Ligand-Enabled γ-C(sp(3))-H Olefination of Amines: En Route to Pyrrolidines.Journal of the American Chemical Society · 2016Article
- The syn/anti-dichotomy in the palladium-catalyzed addition of nucleophiles to alkenes.Chemistry (Weinheim an der Bergstrasse, Germany) · 2015Article
- Mechanistic studies of Wacker-type amidocyclization of alkenes catalyzed by (IMes)Pd(TFA)2(H2O): kinetic and stereochemical implications of proton transfer.The Journal of organic chemistry · 2013Article
- Characterization of DMSO coordination to palladium(II) in solution and insights into the aerobic oxidation catalyst, Pd(DMSO)2(TFA)2.Inorganic chemistry · 2012Article
- Stereoselective synthesis of morpholines via copper-promoted oxyamination of alkenes.Organic letters · 2012Article
Corrections and comments
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Authors and funding
2 authors.
Funding
Abstract
Use of a base-free Pd(DMSO)(2)(TFA)(2) catalyst system enables the synthesis of six-membered nitrogen heterocycles via a Wacker-type aerobic oxidative cyclization of alkenes bearing tethered sulfonamides. Various heterocycles, including morpholines, piperidines, piperazines, and piperazinones, are accessible by this method.
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Registered trials
Read under generation 80e0d062 · epoch 390. Bibliography from PubMed, PubMed Central and OpenAlex; grants from NIH RePORTER; trial links from ClinicalTrials.gov; estimates, votes and beliefs from the OpenQuestion graph.