ArticleOrganic letters2010
General method for synthesis of 2-heterocyclic N-methyliminodiacetic acid boronates.
Article in Organic letters, 2010. The graph could read no effect estimate from its abstract, so it casts no vote on the map. Cited by 22 papers.
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Who cites it
22 citing papers in PubMed.
- A Modular Synthesis of Teraryl-Based α-Helix Mimetics, Part 5: A Complete Set of Pyridine Boronic Acid Pinacol Esters Featuring Side Chains of Proteinogenic Amino Acids.European journal of organic chemistry · 2022Article
- Preparation of MIDA Anhydride and Reaction with Boronic Acids.Organic syntheses; an annual publication of satisfactory methods for the preparation of organic chemicals · 2022Article
- Heteroaryl-Heteroaryl, Suzuki-Miyaura, Anhydrous Cross-Coupling Reactions Enabled by Trimethyl Borate.Journal of the American Chemical Society · 2021Article
- Light-Mediated Cross-Coupling of Anomeric Trifluoroborates.Organic letters · 2021Article
- Synthesis of Tridentate [1,2,4] Triazinyl-Pyridin-2-yl Indole Lewis Basic Complexants via Pd-Catalyzed Suzuki-Miyaura Cross-Coupling.ACS omega · 2019Article
- The Molecular Industrial Revolution: Automated Synthesis of Small Molecules.Angewandte Chemie (International ed. in English) · 2018Review
- Design, Synthesis, and Application of Polymer-Supported Silicon-Transfer Agents for Cross-Coupling Reactions with Organolithium Reagents.The Journal of organic chemistry · 2017Article
- Use ofJournal of polymer science. Part A, Polymer chemistry · 2017Article
- Design, Synthesis, and Validation of an Effective, Reusable Silicon-Based Transfer Agent for Room-Temperature Pd-Catalyzed Cross-Coupling Reactions of Aryl and Heteroaryl Chlorides with Readily Available Aryl Lithium Reagents.Journal of the American Chemical Society · 2016Article
- Ru-catalysed C-H arylation of indoles and pyrroles with boronic acids: scope and mechanistic studies.Chemistry (Weinheim an der Bergstrasse, Germany) · 2015Article
- Facile synthesis of borofragments and their evaluation in activity-based protein profiling.Chemical communications (Cambridge, England) · 2015Article
- Chemoselective boronic ester synthesis by controlled speciation.Angewandte Chemie (International ed. in English) · 2014Article
- Nickel-catalyzed cross-electrophile coupling of 2-chloropyridines with alkyl bromides.Synlett : accounts and rapid communications in synthetic organic chemistry · 2014Article
- (1-bromovinyl)-MIDA boronate: a readily accessible and highly versatile building block for small molecule synthesis.Tetrahedron · 2013Article
- Copper(II)- and palladium(II)-catalyzed enantioselective Claisen rearrangement of allyloxy- and propargyloxy-indoles to quaternary oxindoles and spirocyclic lactones.The Journal of organic chemistry · 2012Article
- Oxidative Heck Reactions using Aryltrifluoroborates and Aryl N-Methyliminodiacetic Acid (MIDA) Boronates.ChemistryOpen · 2012Article
- A general solution for the 2-pyridyl problem.Angewandte Chemie (International ed. in English) · 2012Article
- Asymmetric synthesis of allenyl oxindoles and spirooxindoles by a catalytic enantioselective Saucy-Marbet Claisen rearrangement.Angewandte Chemie (International ed. in English) · 2012Article
- Pinene-derived iminodiacetic acid (PIDA): a powerful ligand for stereoselective synthesis and iterative cross-coupling of C(sp3) boronate building blocks.Journal of the American Chemical Society · 2011Article
- (Z)-(2-bromovinyl)-MIDA boronate: a readily accessible and highly versatile building block for small molecule synthesis.Tetrahedron · 2011Article
Corrections and comments
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Authors and funding
4 authors.
Funding
Abstract
A wide range of 2-pyridyl and other difficult-to-access heterocyclic N-methyliminodiacetic acid boronates can be readily prepared from the corresponding bromides via a new method involving direct transligation of 2-heterocyclic trialkoxyborate salts with N-methyliminodiacetic acid (MIDA) at elevated temperatures.
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